Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50036152
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50212827(CHEMBL3350189)
Affinity DataKi: <1nMAssay Description:Antagonism against bradykinin receptor B2 in guinea pig ileal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231016(CHEMBL409073)
Affinity DataKi: <5nMAssay Description:Tested for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231125(CHEMBL313256)
Affinity DataKi: <5nMAssay Description:Tested for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231130(CHEMBL2304004)
Affinity DataKi: <5nMAssay Description:Antagonism against bradykinin receptor B2 in guinea pig ileal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231126(CHEMBL2304050)
Affinity DataKi: <5nMAssay Description:Antagonism against bradykinin receptor B2 in guinea pig ileal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50422002(CHEMBL2304049)
Affinity DataKi:  8nMAssay Description:Tested for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231128(CHEMBL2304003)
Affinity DataKi: <10nMAssay Description:Antagonism against bradykinin receptor B2 in guinea pig ileal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231017(CHEMBL1790706)
Affinity DataKi: <10nMAssay Description:Tested for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50231127(CHEMBL2304047)
Affinity DataKi: <10nMAssay Description:Selective binding affinity against Opioid receptor delta 1, using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50422001(CHEMBL2304002)
Affinity DataKi:  10nMAssay Description:Tested for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50044556(1N-(2-hydroxy-1H-1-indenyl)-6-cyclohexyl-3,4-dihyd...)
Affinity DataKi:  30nMAssay Description:Tested for inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed