Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 50048912
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231178(CHEMBL75801)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231221(CHEMBL309693)
Affinity DataEC50:  4.10E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231180(CHEMBL80199)
Affinity DataEC50:  4.58E+3nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231181(CHEMBL80637)
Affinity DataEC50:  360nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231182(CHEMBL80456)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231183(CHEMBL80533)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231184(CHEMBL80692)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231185(CHEMBL76731)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231186(CHEMBL309891)
Affinity DataEC50:  110nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231187(CHEMBL79105)
Affinity DataEC50:  2.10E+4nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  300nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231188(CHEMBL80744)
Affinity DataEC50:  7.77E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231189(CHEMBL80200)
Affinity DataEC50:  1.96E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  300nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231190(CHEMBL80157)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231191(CHEMBL75701)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231192(CHEMBL306733)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231193(CHEMBL79119)
Affinity DataEC50:  2.65E+4nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231194(CHEMBL77231)
Affinity DataEC50:  8.10E+3nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231195(CHEMBL77089)
Affinity DataEC50:  1.08E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231196(CHEMBL77299)
Affinity DataEC50:  5.01E+4nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231197(CHEMBL78616)
Affinity DataEC50:  160nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231166(CHEMBL58719)
Affinity DataEC50:  60nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231198(CHEBI:46932 | Dihydrocapsaicin)
Affinity DataEC50:  190nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231199(CHEMBL80858)
Affinity DataEC50:  3.09E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231200(CHEMBL77292)
Affinity DataEC50:  350nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231201(CHEMBL309762)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231202(CHEMBL80404)
Affinity DataEC50:  290nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231203(CHEMBL309532)
Affinity DataEC50:  180nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231204(CHEMBL80662)
Affinity DataEC50:  100nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50044767(CHEMBL75124 | Hydroxymethoxybenzyl pelargonamide |...)
Affinity DataEC50:  550nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231205(CHEMBL77748)
Affinity DataEC50:  7.98E+4nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231206(CHEMBL76196)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231207(CHEMBL309275)
Affinity DataEC50:  620nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231208(CHEMBL76305)
Affinity DataEC50:  1.00E+6nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231209(CHEMBL77195)
Affinity DataEC50:  1.18E+4nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231210(CHEMBL76571)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231211(CHEMBL309190)
Affinity DataEC50:  4.39E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231212(CHEMBL79767)
Affinity DataEC50:  4.20E+3nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231213(CHEMBL310591)
Affinity DataEC50:  660nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231214(CHEMBL311678)
Affinity DataEC50:  9.48E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231215(CHEMBL80341)
Affinity DataEC50:  1.24E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231216(CHEMBL78895)
Affinity DataEC50:  240nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231217(CHEMBL78533)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231218(CHEMBL76848)
Affinity DataEC50:  270nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231219(CHEMBL80415)
Affinity DataEC50:  2.58E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM20460((9Z)-N-[(4-hydroxy-3-methoxyphenyl)methyl]octadec-...)
Affinity DataEC50:  170nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231220(CHEMBL78640)
Affinity DataEC50:  4.53E+4nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50231179(CHEMBL80495)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed