Affinity DataIC50: 1nMAssay Description:Inhibitory activity against mu-opioid receptor in guinea pig ileum longitudinal muscle using morphineMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against delta-opioid receptor in mouse vas deferens preparation using DADLEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against kappa-opioid receptor in guinea pig ileum longitudinal muscle using ethylketazocineMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against mu-opioid receptor in guinea pig ileum longitudinal muscle using morphineMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibitory activity against mu-opioid receptor in guinea pig ileum longitudinal muscle using morphineMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Inhibitory activity against delta-opioid receptor in mouse vas deferens preparation using DADLEMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against delta-opioid receptor in mouse vas deferens preparation using DADLEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against kappa-opioid receptor in guinea pig ileum longitudinal muscle using ethylketazocineMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 181nMAssay Description:Inhibitory activity against kappa-opioid receptor in guinea pig ileum longitudinal muscle using ethylketazocineMore data for this Ligand-Target Pair