Compile Data Set for Download or QSAR
maximum 50k data
Found 67 Enz. Inhib. hit(s) with all data for entry = 50006185
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045797(2-[3-(4-Chloro-phenyl)-ureido]-3-(1H-indol-3-yl)-2...)
Affinity DataKi: >0.000100nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  6.10nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  6.5nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  12nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  14nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in mouse brain by displacement of [3H]-pBC264 radioligand (icv)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  14nMAssay Description:Tested for binding affinity towards cholecystokinin type A receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  14nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  18nMAssay Description:Tested for binding affinity towards CCK-B in rat cortex by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  21nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in rat cortex by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  21nMAssay Description:Tested for binding affinity towards CCK-B in mouse brain by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045798(CHEMBL319120 | [1-[2-(2,4-Dichloro-phenyl)-ethylca...)
Affinity DataKi:  27nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  28nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045810(3-{[2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol...)
Affinity DataKi:  36nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045816(CHEMBL319880 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  37nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045803(CHEMBL433407 | [1-[2-(4-Chloro-phenyl)-ethylcarbam...)
Affinity DataKi:  39nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  40nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in rat cortex by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045806(CHEMBL320399 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  50nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045808(CHEMBL432389 | [1-[2-(4-Bromo-phenyl)-ethylcarbamo...)
Affinity DataKi:  51nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045802(CHEMBL99252 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  70nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  73nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in mouse brain by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045813(CHEMBL328852 | {2-(1H-Indol-3-yl)-1-methyl-1-[2-(4...)
Affinity DataKi:  79nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045817(CHEMBL319085 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  87nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50005823(CHEMBL291033 | [2-(1H-Indol-3-yl)-1-methyl-1-phene...)
Affinity DataKi:  87nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045818(CHEMBL95115 | [2-(1H-Indol-3-yl)-1-methyl-1-(2-nap...)
Affinity DataKi:  89nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045804(CHEMBL329088 | {2-(1H-Indol-3-yl)-1-[2-(4-methoxy-...)
Affinity DataKi:  115nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045815(CHEMBL98516 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  134nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045814(CHEMBL95793 | [2-(1H-Indol-3-yl)-1-methyl-1-(3-phe...)
Affinity DataKi:  182nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045809(CHEMBL316462 | [1-[2-(3,4-Dichloro-phenyl)-ethylca...)
Affinity DataKi:  184nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045801(CHEMBL95461 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  224nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045812(CHEMBL99076 | [1-Benzylcarbamoyl-2-(1H-indol-3-yl)...)
Affinity DataKi:  231nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045819(CHEMBL95689 | [2-(1H-Indol-3-yl)-1-methyl-1-(napht...)
Affinity DataKi:  402nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045799(CHEMBL318238 | [2-(1H-Indol-3-yl)-1-methyl-1-pheny...)
Affinity DataKi:  407nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  531nMAssay Description:Tested for binding affinity towards cholecystokinin type A receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045821(CHEMBL320823 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  543nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045820(3-(1H-Indol-3-yl)-2-methyl-2-(3-naphthalen-2-yl-ur...)
Affinity DataKi:  769nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045811(CHEMBL96036 | [2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  986nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045816(CHEMBL319880 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  1.04E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  1.06E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  1.13E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  1.22E+3nMAssay Description:Tested for binding affinity towards cholecystokinin type A receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  1.23E+3nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in mouse brain by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045810(3-{[2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol...)
Affinity DataKi:  1.32E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  1.36E+3nMAssay Description:Tested for binding affinity towards cholecystokinin type A receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  1.52E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045809(CHEMBL316462 | [1-[2-(3,4-Dichloro-phenyl)-ethylca...)
Affinity DataKi:  1.54E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045803(CHEMBL433407 | [1-[2-(4-Chloro-phenyl)-ethylcarbam...)
Affinity DataKi:  1.61E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045807(3-(1H-Indol-3-yl)-2-methyl-N-phenethyl-2-(3-trityl...)
Affinity DataKi:  1.78E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50005823(CHEMBL291033 | [2-(1H-Indol-3-yl)-1-methyl-1-phene...)
Affinity DataKi:  1.89E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045815(CHEMBL98516 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  2.01E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045808(CHEMBL432389 | [1-[2-(4-Bromo-phenyl)-ethylcarbamo...)
Affinity DataKi:  2.14E+3nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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