Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50006285
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047064(4-[5-Fluoro-1-(4-methoxy-benzyl)-1H-benzoimidazol-...)
Affinity DataKi:  4nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047082(4-[5-Fluoro-1-(4-methylsulfanyl-benzyl)-1H-benzoim...)
Affinity DataKi:  5nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047054(4-[1-(3,4-Dichloro-benzyl)-5-fluoro-1H-benzoimidaz...)
Affinity DataKi:  6nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047068(4-[5-Chloro-1-(4-methylsulfanyl-benzyl)-1H-benzoim...)
Affinity DataKi:  6nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047081(4-[6-Chloro-3-(4-methylsulfanyl-benzyl)-3H-imidazo...)
Affinity DataKi:  7nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047065(4-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  7.80nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047058(4-[1-(4-Bromo-2-fluoro-benzyl)-1H-benzoimidazol-2-...)
Affinity DataKi:  11nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047059(4-[5-Chloro-1-(3,4-dichloro-benzyl)-1H-benzoimidaz...)
Affinity DataKi:  12nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047076(4-[1-(4-Bromo-benzyl)-5-fluoro-1H-benzoimidazol-2-...)
Affinity DataKi:  12nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047072(4-[1-(4-Bromo-benzyl)-5-chloro-1H-benzoimidazol-2-...)
Affinity DataKi:  13nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047067(4-[1-(4-Bromo-2-fluoro-benzyl)-5-fluoro-1H-benzoim...)
Affinity DataKi:  15nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50008779((+) [9-(4-Chloro-benzyl)-6-fluoro-2,3,4,9-tetrahyd...)
Affinity DataKi:  15.3nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047079(4-[1-(4-Bromo-benzyl)-1H-benzoimidazol-2-yl]-3,3-d...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047083(4-[5-Chloro-1-(4-methoxy-benzyl)-1H-benzoimidazol-...)
Affinity DataKi:  20nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047060(4-[6-Chloro-3-(4-chloro-benzyl)-3H-imidazo[4,5-b]p...)
Affinity DataKi:  21nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047066(4-[5-Chloro-1-(4-chloro-benzyl)-1H-benzoimidazol-2...)
Affinity DataKi:  23nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047062(5-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  23nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047077(4-[1-(4-Chloro-benzyl)-1H-benzoimidazol-2-yl]-3,3-...)
Affinity DataKi:  31nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047063(4-[1-(4-Methoxy-benzyl)-1H-benzoimidazol-2-yl]-3,3...)
Affinity DataKi:  31nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047055(4-[5-Fluoro-1-(4-methanesulfonyl-benzyl)-1H-benzoi...)
Affinity DataKi:  37nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047080(4-[3-(4-Chloro-benzyl)-3H-imidazo[4,5-b]pyridin-2-...)
Affinity DataKi:  39nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047078(CHEMBL18206 | {1-[1-(4-Chloro-benzyl)-5-fluoro-1H-...)
Affinity DataKi:  42nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047075(CHEMBL18232 | {1-[1-(4-Chloro-benzyl)-5-fluoro-1H-...)
Affinity DataKi:  52nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047074(3,3-Dimethyl-4-[1-(4-nitro-benzyl)-1H-benzoimidazo...)
Affinity DataKi:  60nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047073(2-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  140nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047053(3-[1-(4-Chloro-benzyl)-1H-benzoimidazol-2-ylmethyl...)
Affinity DataKi:  160nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047071(6-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  510nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50002765(BM 13177 | BM-13177 | CHEMBL8273 | Sulotroban | [4...)
Affinity DataKi:  650nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047056(2-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  670nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047057(2-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  810nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047069(CHEMBL275651 | {1-[1-(4-Chloro-benzyl)-5-fluoro-1H...)
Affinity DataKi:  870nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047061(3-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  1.70E+3nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50047070(3-[1-(4-Chloro-benzyl)-5-fluoro-1H-benzoimidazol-2...)
Affinity DataKi:  5.60E+3nMAssay Description:Tested in vitro for inhibition constant against TXA2 / PGH-2 receptor using [125I]-PTA-OH binding affinity to human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed