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Found 38 Enz. Inhib. hit(s) with all data for entry = 50006458
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049365(1-Benzyl-4-{2-[bis-(4-fluoro-phenyl)-methoxy]-ethy...)
Affinity DataIC50:  9.70nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049360(4-(2-Benzhydryloxy-ethyl)-1-phenethyl-piperidine |...)
Affinity DataIC50:  10.6nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049359(4-(2-Benzhydryloxy-ethyl)-1-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  12nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049371(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-(3-pheny...)
Affinity DataIC50:  13nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049364(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-phenethy...)
Affinity DataIC50:  13.5nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049369(4-Benzhydryloxymethyl-1-(3-phenyl-propyl)-piperidi...)
Affinity DataIC50:  14.5nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049362(4-(2-Benzhydryloxy-ethyl)-1-benzyl-piperidine | CH...)
Affinity DataIC50:  15.2nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049363(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50:  16.7nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049357(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50:  19.9nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049357(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50:  31.9nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049363(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50:  55nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049369(4-Benzhydryloxymethyl-1-(3-phenyl-propyl)-piperidi...)
Affinity DataIC50:  58nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049372(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50:  65nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataIC50:  82nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049360(4-(2-Benzhydryloxy-ethyl)-1-phenethyl-piperidine |...)
Affinity DataIC50:  102nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049358(4-Benzhydryloxymethyl-1-phenethyl-piperidine | CHE...)
Affinity DataIC50:  108nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049371(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-(3-pheny...)
Affinity DataIC50:  112nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049367(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50:  115nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049373(1-Benzyl-4-[bis-(4-fluoro-phenyl)-methoxymethyl]-p...)
Affinity DataIC50:  126nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049368(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-(3-ph...)
Affinity DataIC50:  159nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049365(1-Benzyl-4-{2-[bis-(4-fluoro-phenyl)-methoxy]-ethy...)
Affinity DataIC50:  198nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049372(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataIC50:  224nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049359(4-(2-Benzhydryloxy-ethyl)-1-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  232nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049364(4-[Bis-(4-fluoro-phenyl)-methoxymethyl]-1-phenethy...)
Affinity DataIC50:  237nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049361(4-{2-[Bis-(4-methoxy-phenyl)-methoxy]-ethyl}-1-(3-...)
Affinity DataIC50:  255nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049374(4-(2-Di-p-tolylmethoxy-ethyl)-1-phenethyl-piperidi...)
Affinity DataIC50:  311nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049361(4-{2-[Bis-(4-methoxy-phenyl)-methoxy]-ethyl}-1-(3-...)
Affinity DataIC50:  340nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049366(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-phene...)
Affinity DataIC50:  382nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049367(4-{2-[Bis-(4-chloro-phenyl)-methoxy]-ethyl}-1-phen...)
Affinity DataIC50:  414nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049358(4-Benzhydryloxymethyl-1-phenethyl-piperidine | CHE...)
Affinity DataIC50:  456nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049370(4-Benzhydryloxymethyl-1-benzyl-piperidine | CHEMBL...)
Affinity DataIC50:  544nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049366(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-phene...)
Affinity DataIC50:  638nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049370(4-Benzhydryloxymethyl-1-benzyl-piperidine | CHEMBL...)
Affinity DataIC50:  702nMAssay Description:Binding affinity at dopamine transporter from rat striatal membrane tissue by [3H]-CFT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049362(4-(2-Benzhydryloxy-ethyl)-1-benzyl-piperidine | CH...)
Affinity DataIC50:  743nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049373(1-Benzyl-4-[bis-(4-fluoro-phenyl)-methoxymethyl]-p...)
Affinity DataIC50:  761nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049368(4-{2-[Bis-(4-bromo-phenyl)-methoxy]-ethyl}-1-(3-ph...)
Affinity DataIC50:  835nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50049374(4-(2-Di-p-tolylmethoxy-ethyl)-1-phenethyl-piperidi...)
Affinity DataIC50:  888nMAssay Description:Binding affinity at serotonin transporter from rat brain striatal membrane by [3H]-citalopram displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed