Affinity DataKi: 0.75nMAssay Description:Binding affinity against Opioid receptor mu 1 in Guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.980nMAssay Description:Binding affinity against Opioid receptor mu 1 in Guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.24nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Binding affinity against Opioid receptor kappa 1 in Guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranes using [3H]DAMGO+DADLEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Binding affinity against Kappa Opioid receptor in Guinea pig brain membranes using [3H]-DAMGO+EKCMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Binding affinity against Kappa Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 183nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Opioid receptor mu 1 antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Opioid receptor mu 1 antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair