Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50036504
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  0.75nMAssay Description:Binding affinity against Opioid receptor mu 1 in Guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049563(5-amino-2,4(Bis-4-cyclopropylmethyl-10,17-dihydrox...)
Affinity DataKi:  0.980nMAssay Description:Binding affinity against Opioid receptor mu 1 in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049560((4S,5'R,13'R,17'S)-2-[(5R,13R,14R,17S)-14-amino-4-...)
Affinity DataKi:  1.24nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049560((4S,5'R,13'R,17'S)-2-[(5R,13R,14R,17S)-14-amino-4-...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity against Opioid receptor kappa 1 in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  20nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranes using [3H]DAMGO+DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  36nMAssay Description:Binding affinity against Kappa Opioid receptor in Guinea pig brain membranes using [3H]-DAMGO+EKCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049563(5-amino-2,4(Bis-4-cyclopropylmethyl-10,17-dihydrox...)
Affinity DataKi:  88nMAssay Description:Binding affinity against Kappa Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049563(5-amino-2,4(Bis-4-cyclopropylmethyl-10,17-dihydrox...)
Affinity DataKi:  183nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049564(14-amino-14-amino(imino)methyl-4-cyclopropylmethyl...)
Affinity DataIC50:  18nMAssay Description:Opioid receptor mu 1 antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50049561(CHEMBL430950 | Naltrexone derivative)
Affinity DataIC50:  71nMAssay Description:Opioid receptor mu 1 antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed