Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50006492
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50454480(CHEMBL2093059)
Affinity DataIC50:  0.0540nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50454481(CHEMBL2110201)
Affinity DataIC50:  0.0740nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049783(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049789(1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50454482(CHEMBL2110202)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049785(1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049786(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  0.580nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049788(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049790(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049784(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049787(1-{4-Methyl-3-[methyl-(1H-tetrazol-5-yl)-amino]-ph...)
Affinity DataIC50:  20nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50454482(CHEMBL2110202)
Affinity DataIC50:  153nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049789(1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50454480(CHEMBL2093059)
Affinity DataIC50:  400nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  736nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50454481(CHEMBL2110201)
Affinity DataIC50:  802nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049785(1-((R)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049790(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049786(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049787(1-{4-Methyl-3-[methyl-(1H-tetrazol-5-yl)-amino]-ph...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049788(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049784(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049783(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  4.08E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed