Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50036424
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407836(CHEMBL2112240)
Affinity DataIC50:  2nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407838(CHEMBL2112243)
Affinity DataIC50:  15nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407835(CHEMBL2112242)
Affinity DataIC50:  28nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407839(CHEMBL2112244)
Affinity DataIC50:  35nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407840(CHEMBL2112241)
Affinity DataIC50:  59nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051573(CHEMBL420221 | N-(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-b...)
Affinity DataIC50:  60nMAssay Description:Binding affinity towards Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369144(CHEMBL2369607)
Affinity DataIC50:  85nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407834(CHEMBL2092730)
Affinity DataIC50:  95nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataIC50:  180nMAssay Description:Binding affinity towards Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369141(CHEMBL2369606)
Affinity DataIC50:  198nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50407837(CHEMBL2092883)
Affinity DataIC50:  496nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369133(CHEMBL2369601)
Affinity DataIC50:  549nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369136(CHEMBL2369604)
Affinity DataIC50:  596nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369143(CHEMBL1790623)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369134(CHEMBL2369600)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369132(CHEMBL2369603)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369138(CHEMBL2369605)
Affinity DataIC50:  2.73E+3nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051578(5-{(2R,3S,5R,6R)-3,5-Bis-benzyloxy-6-[2-(1H-indol-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding affinity towards cloned human Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding affinity towards cloned human Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369139(CHEMBL2369599)
Affinity DataIC50:  4.09E+3nMAssay Description:Inhibition of Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataIC50:  1.20E+5nMAssay Description:Binding affinity towards Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed