Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50041250
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408044(CHEMBL3038104)
Affinity DataIC50:  1.62E+3nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408047(CHEMBL3038096)
Affinity DataIC50:  3.02E+3nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408048(CHEMBL3038099)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408052(CHEMBL3038097)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408058(CHEMBL2028982)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408053(CHEMBL3038094)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408055(CHEMBL3038102)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Cortech

Curated by ChEMBL
LigandPNGBDBM50408049(CHEMBL3038098)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408053(CHEMBL3038094)
Affinity DataKd:  3.16nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408044(CHEMBL3038104)
Affinity DataKd:  174nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408045(CHEMBL2372278)
Affinity DataKd:  0.490nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408055(CHEMBL3038102)
Affinity DataKd:  50.1nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408047(CHEMBL3038096)
Affinity DataKd:  18.6nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed