Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50006667
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM8903((1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltet...)
Affinity DataIC50:  30nMAssay Description:Inhibition of 10e-9 M aldosterone activity in CV-1 cells expressing mineralocorticoid receptorMore data for this Ligand-Target Pair
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50407855(CHEMBL2112397)
Affinity DataIC50:  700nMAssay Description:Inhibition of 10e-9 M aldosterone activity in CV-1 cells expressing mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50407856(CHEMBL2112398)
Affinity DataIC50:  900nMAssay Description:Inhibition of 10e-9 M aldosterone activity in CV-1 cells expressing mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50422147(CHEMBL97531)
Affinity DataKd:  0.740nMAssay Description:Affinity for recombinant Mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50407856(CHEMBL2112398)
Affinity DataKd:  20nMAssay Description:Affinity for recombinant Mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50407855(CHEMBL2112397)
Affinity DataKd:  20nMAssay Description:Affinity for recombinant Mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM8903((1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltet...)
Affinity DataKd:  0.390nMAssay Description:Affinity for recombinant Mineralocorticoid receptorMore data for this Ligand-Target Pair