Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50006952
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056102((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056093(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056103(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056099(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056092(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50:  0.140nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056091(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50:  0.160nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056089(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056095(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056098(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50:  0.210nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056086(1-(3-Amino-phenyl)-3-[(R)-1-(3,3-dimethyl-2-oxo-bu...)
Affinity DataIC50:  0.430nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056096(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  0.440nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056094(1-(3-Amino-phenyl)-3-[(R)-1-(3,3-dimethyl-2-oxo-bu...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  0.520nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056085(CHEMBL325746 | N-(3-{3-[1-(3,3-Dimethyl-2-oxo-buty...)
Affinity DataIC50:  0.590nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056100(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  0.840nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056090(1-(3-Dimethylamino-phenyl)-3-[(S)-1-(3,3-dimethyl-...)
Affinity DataIC50:  1.26nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056088(1-(3-Cyano-phenyl)-3-[1-(3,3-dimethyl-2-oxo-butyl)...)
Affinity DataIC50:  1.29nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056087(3-{3-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-...)
Affinity DataIC50:  3.29nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056098(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50:  89nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  111nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056095(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50:  113nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056093(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataIC50:  146nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056089(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50:  157nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056099(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  253nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056103(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50:  301nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056096(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  470nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056102((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...)
Affinity DataIC50:  502nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056092(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50:  558nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056085(CHEMBL325746 | N-(3-{3-[1-(3,3-Dimethyl-2-oxo-buty...)
Affinity DataIC50:  561nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056090(1-(3-Dimethylamino-phenyl)-3-[(S)-1-(3,3-dimethyl-...)
Affinity DataIC50:  572nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056091(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50:  589nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056088(1-(3-Cyano-phenyl)-3-[1-(3,3-dimethyl-2-oxo-butyl)...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056100(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50:  944nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056094(1-(3-Amino-phenyl)-3-[(R)-1-(3,3-dimethyl-2-oxo-bu...)
Affinity DataIC50:  953nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056086(1-(3-Amino-phenyl)-3-[(R)-1-(3,3-dimethyl-2-oxo-bu...)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056087(3-{3-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-...)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed