Affinity DataKi: 0.650nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at Adenosine A2A receptor in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 169nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 198nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 296nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 305nMAssay Description:Displacement of specific [3H]-(R)-PIA binding at adenosine A1 receptor from rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 314nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 443nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 507nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 567nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.38E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.42E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.52E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.69E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.72E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.27E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.44E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.58E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 2.74E+3nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at Adenosine A2A receptor in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of specific [125I]-AB-MECA binding at rat Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair