Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50007215
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059767((2R,6S,11R)-3-((S)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059778((2R,6S)-3-((S)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059761((2R,6S,11R)-6,11-Dimethyl-3-((S)-2-methylsulfanyl-...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059772((2R,6S,11S)-3-((S)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059764((2R,6S,11R)-3-(2-Methoxy-2-methyl-propyl)-6,11-dim...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059786((2R,6S,11R)-6,11-Dimethyl-3-((R)-2-methylsulfanyl-...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059800((2R,6S)-3-((S)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  18.2nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059794((2R,6R)-3-((S)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  20.9nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059803((2R,6S,11S)-6,11-Dimethyl-3-((S)-2-methylsulfanyl-...)
Affinity DataKi:  97nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059783((2R,6S)-3-((R)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  108nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059788((2R,6S)-3-((S)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  144nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059766((2R,6S,11R)-3-((R)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  146nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059792((2R,6S,11S)-3-((R)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  212nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059797((2R,6S,11S)-6,11-Dimethyl-3-((R)-2-methylsulfanyl-...)
Affinity DataKi:  236nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059771((2S,6R)-3-((S)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059777((2R,6S)-3-((R)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059782((2S,6R,11S)-3-((S)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059759((2S,6R)-3-((S)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  6.02E+3nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059770((2R,6R)-3-((R)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  1.14E+4nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059776((2S,6R)-3-((R)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059774((2S,6R,11S)-3-((R)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  1.84E+4nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059773((2S,6R,11R)-3-((R)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  3.48E+4nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059763((2R,6S)-3-((R)-2-Methoxy-propyl)-6,11,11-trimethyl...)
Affinity DataKi:  4.24E+4nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50059768((2S,6R,11R)-3-((S)-2-Methoxy-propyl)-6,11-dimethyl...)
Affinity DataKi:  6.66E+4nMAssay Description:Inhibition of [3H]-dihydromorphine binding to opioid receptor mu 1 in rat brain cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed