Compile Data Set for Download or QSAR
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Found 55 Enz. Inhib. hit(s) with all data for entry = 50007372
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062027(3-(3-Carbamimidoyl-phenyl)-5-(4-guanidino-phenyl)-...)
Affinity DataKi:  9nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062035(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  34nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062033(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  42nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062038(3-(3-Carbamimidoyl-phenyl)-7-(4-guanidino-phenyl)-...)
Affinity DataKi:  57nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062027(3-(3-Carbamimidoyl-phenyl)-5-(4-guanidino-phenyl)-...)
Affinity DataKi:  96nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062035(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  99nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062031(3-(3-Carbamimidoyl-phenyl)-5-(4-methanesulfonylami...)
Affinity DataKi:  110nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062033(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  110nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062024(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  140nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062024(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  192nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062019(4-[3-(3-Carbamimidoyl-phenyl)-4-methoxycarbonyl-bu...)
Affinity DataKi:  330nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062037(3-[3-amino(imino)methylphenyl]-5-[4-amino(imino)me...)
Affinity DataKi:  440nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062034(3-(3-Carbamimidoyl-phenyl)-5-(4-carbamoyl-phenyl)-...)
Affinity DataKi:  550nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062023(5-(4-Benzenesulfonylamino-phenyl)-3-(3-carbamimido...)
Affinity DataKi:  610nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062031(3-(3-Carbamimidoyl-phenyl)-5-(4-methanesulfonylami...)
Affinity DataKi:  654nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062038(3-(3-Carbamimidoyl-phenyl)-7-(4-guanidino-phenyl)-...)
Affinity DataKi:  760nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062036(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  820nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062034(3-(3-Carbamimidoyl-phenyl)-5-(4-carbamoyl-phenyl)-...)
Affinity DataKi:  870nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062036(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  940nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062023(5-(4-Benzenesulfonylamino-phenyl)-3-(3-carbamimido...)
Affinity DataKi:  1.10E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062033(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  1.10E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062037(3-[3-amino(imino)methylphenyl]-5-[4-amino(imino)me...)
Affinity DataKi:  1.15E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062022(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi: >1.20E+3nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062035(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  1.20E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062026(5-(4-Amino-phenyl)-3-(3-carbamimidoyl-phenyl)-pent...)
Affinity DataKi:  1.20E+3nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062020(3,5-Bis-(4-carbamimidoyl-phenyl)-pentanoic acid et...)
Affinity DataKi:  1.20E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062022(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062024(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  1.54E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062028(5-(3-Carbamimidoyl-phenyl)-3-(4-carbamimidoyl-phen...)
Affinity DataKi:  1.64E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062023(5-(4-Benzenesulfonylamino-phenyl)-3-(3-carbamimido...)
Affinity DataKi:  1.75E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062021(3-(3-Carbamimidoyl-phenyl)-5-phenyl-pentanoic acid...)
Affinity DataKi: >2.10E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062029(CHEMBL155632 | [5-(4-Carbamimidoyl-phenyl)-3-(3-ca...)
Affinity DataKi:  2.40E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062025(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  2.40E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062019(4-[3-(3-Carbamimidoyl-phenyl)-4-methoxycarbonyl-bu...)
Affinity DataKi:  2.80E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062039(3,5-Bis-(3-carbamimidoyl-phenyl)-pentanoic acid me...)
Affinity DataKi:  2.80E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062037(3-[3-amino(imino)methylphenyl]-5-[4-amino(imino)me...)
Affinity DataKi:  2.80E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062021(3-(3-Carbamimidoyl-phenyl)-5-phenyl-pentanoic acid...)
Affinity DataKi:  2.90E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062031(3-(3-Carbamimidoyl-phenyl)-5-(4-methanesulfonylami...)
Affinity DataKi:  3.10E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062027(3-(3-Carbamimidoyl-phenyl)-5-(4-guanidino-phenyl)-...)
Affinity DataKi:  3.10E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062038(3-(3-Carbamimidoyl-phenyl)-7-(4-guanidino-phenyl)-...)
Affinity DataKi:  3.30E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062028(5-(3-Carbamimidoyl-phenyl)-3-(4-carbamimidoyl-phen...)
Affinity DataKi:  3.43E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062019(4-[3-(3-Carbamimidoyl-phenyl)-4-methoxycarbonyl-bu...)
Affinity DataKi:  3.60E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062022(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi: >4.20E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062030(1-[3-amino(imino)methylphenyl]-3-[4-amino(imino)me...)
Affinity DataKi:  4.40E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062026(5-(4-Amino-phenyl)-3-(3-carbamimidoyl-phenyl)-pent...)
Affinity DataKi:  5.00E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062030(1-[3-amino(imino)methylphenyl]-3-[4-amino(imino)me...)
Affinity DataKi:  5.10E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062032(5-(4-Carbamimidoyl-phenyl)-3-phenyl-pentanoic acid...)
Affinity DataKi:  6.20E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062034(3-(3-Carbamimidoyl-phenyl)-5-(4-carbamoyl-phenyl)-...)
Affinity DataKi:  6.50E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062026(5-(4-Amino-phenyl)-3-(3-carbamimidoyl-phenyl)-pent...)
Affinity DataKi:  7.70E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062036(5-(4-Carbamimidoyl-phenyl)-3-(3-carbamimidoyl-phen...)
Affinity DataKi:  8.00E+3nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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