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Found 26 Enz. Inhib. hit(s) with all data for entry = 3602
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36643(L-161,189)
Affinity DataIC50:  300nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36644(L-159,906)
Affinity DataIC50:  400nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36639(L-158-817)
Affinity DataIC50:  1.80E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36640(CHEMBL26514 | L-159,061)
Affinity DataIC50:  1.90E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36638(L-158-678)
Affinity DataIC50:  3.50E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36636(L-809-559)
Affinity DataIC50:  4.00E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36642(L-809,370)
Affinity DataIC50:  6.00E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50:  7.00E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36641(L-809,339)
Affinity DataIC50:  4.20E+4nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36637(L-809-558)
Affinity DataIC50:  4.20E+4nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36644(L-159,906)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36642(L-809,370)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36641(L-809,339)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36640(CHEMBL26514 | L-159,061)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36639(L-158-817)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36635(L-808,509)
Affinity DataIC50:  1.10E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36643(L-161,189)
Affinity DataIC50:  1.20E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36634(L-158,507)
Affinity DataIC50:  1.60E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50:  1.90E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36638(L-158-678)
Affinity DataIC50:  2.40E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36637(L-809-558)
Affinity DataIC50: >2.50E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36636(L-809-559)
Affinity DataIC50: >2.50E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36635(L-808,509)
Affinity DataIC50: >5.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36633(L-809,022)
Affinity DataIC50:  8.60E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36634(L-158,507)
Affinity DataIC50: >1.00E+6nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36633(L-809,022)
Affinity DataIC50: >1.00E+6nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed