Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50036619
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064657(CHEMBL277390 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe...)
Affinity DataKi:  85nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (dipeptidylpeptidase 4) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064657(CHEMBL277390 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe...)
Affinity DataKi:  470nMAssay Description:Inhibitory kinetic constant against Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064660(CHEMBL302602 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064657(CHEMBL277390 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064661(CHEMBL67679 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SBu2...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064656(CHEMBL67680 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SOct...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064661(CHEMBL67679 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SBu2...)
Affinity DataIC50:  570nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064660(CHEMBL302602 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe...)
Affinity DataIC50:  610nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064656(CHEMBL67680 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SOct...)
Affinity DataIC50:  630nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064657(CHEMBL277390 | Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2SMe...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064658(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2OAc]-Gly2-), CF3CO...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064658(Cyclo(Lys(alphaH2+)-Pro-Aba-[CH2OAc]-Gly2-), CF3CO...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064659((4S,10S)-10-Amino-24-phenoxymethyl-2,8,15,18,21-pe...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by CD26 (Dipeptidyl peptidase IV) purified from CEM H01 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50064659((4S,10S)-10-Amino-24-phenoxymethyl-2,8,15,18,21-pe...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity against hydrolysis of Gly-Pro-pNa by Dipeptidyl peptidase IV purified from CD26-negative C8166 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed