Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50007599
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065173((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  8nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065188((S)-N-(2-Cyclohexyl-ethyl)-3-{2-[ethyl-(4-piperidi...)
Affinity DataIC50:  10nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065177((S)-N-[(S)-1-Carboxy-2-(decahydro-naphthalen-1-yl)...)
Affinity DataIC50:  11nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065174((S)-N-((R)-1-Carboxy-3-cyclohexyl-propyl)-3-{2-[et...)
Affinity DataIC50:  11nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065185((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065167((S)-N-((R)-2-Cyclohexyl-1-ethoxycarbonyl-ethyl)-3-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50:  17nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065177((S)-N-[(S)-1-Carboxy-2-(decahydro-naphthalen-1-yl)...)
Affinity DataIC50:  19nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065182((S)-N-((S)-1-Carboxy-2-naphthalen-1-yl-ethyl)-3-{2...)
Affinity DataIC50:  22nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065172((S)-N-((S)-1-Carboxy-2-naphthalen-2-yl-ethyl)-3-{2...)
Affinity DataIC50:  22nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50:  26nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065173((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  27nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065166((S)-N-((R)-1-Carbamoyl-2-cyclohexyl-ethyl)-3-{2-[e...)
Affinity DataIC50:  28nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065174((S)-N-((R)-1-Carboxy-3-cyclohexyl-propyl)-3-{2-[et...)
Affinity DataIC50:  31nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065180((S)-N-((R)-Carboxy-cyclohexyl-methyl)-3-{2-[ethyl-...)
Affinity DataIC50:  32nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065186((S)-N-((R)-1-Carboxy-2-cycloheptyl-ethyl)-3-{2-[et...)
Affinity DataIC50:  32nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065181((S)-N-((R)-1-Carboxy-2-cyclopentyl-ethyl)-3-{2-[et...)
Affinity DataIC50:  47nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065184((R)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  53nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065178((S)-N-((S)-1-Carboxy-2-phenyl-ethyl)-3-{2-[ethyl-(...)
Affinity DataIC50:  64nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065167((S)-N-((R)-2-Cyclohexyl-1-ethoxycarbonyl-ethyl)-3-...)
Affinity DataIC50:  64nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065172((S)-N-((S)-1-Carboxy-2-naphthalen-2-yl-ethyl)-3-{2...)
Affinity DataIC50:  68nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065168((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  72nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065188((S)-N-(2-Cyclohexyl-ethyl)-3-{2-[ethyl-(4-piperidi...)
Affinity DataIC50:  72nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065176((S)-N-((R)-1-Carboxy-2-cyclooctyl-ethyl)-3-{2-[eth...)
Affinity DataIC50:  78nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065168((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  82nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065183((S)-N-[(S)-1-Carboxy-2-(decahydro-naphthalen-2-yl)...)
Affinity DataIC50:  96nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065166((S)-N-((R)-1-Carbamoyl-2-cyclohexyl-ethyl)-3-{2-[e...)
Affinity DataIC50:  97nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065182((S)-N-((S)-1-Carboxy-2-naphthalen-1-yl-ethyl)-3-{2...)
Affinity DataIC50:  110nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065190((S)-N-((R)-2-Cyclohexyl-1-hydroxymethyl-ethyl)-3-{...)
Affinity DataIC50:  129nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065185((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  130nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065192((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(5-piperidin-4-yl...)
Affinity DataIC50:  210nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065169((R)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  260nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065165((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(6-guanidino-hexa...)
Affinity DataIC50:  470nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065187((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(5-guanidino-pent...)
Affinity DataIC50:  630nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065169((R)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50:  720nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065189((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(3-piperidin-4-yl...)
Affinity DataIC50:  770nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065170((S)-2-{(S)-3-Carboxy-2-[2-(4-piperidin-4-yl-butyry...)
Affinity DataIC50:  1.06E+3nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065191((S)-N-((R)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50:  1.37E+3nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065179((S)-2-{(S)-3-Carboxy-2-[2-(5-guanidino-pentanoylam...)
Affinity DataIC50:  2.30E+3nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065175(1-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl-but...)
Affinity DataIC50:  3.41E+3nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180((6S,12S,15S)-1,6-diamino-12-(carboxymethyl)-16-hyd...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241181((2S)-2-[(2S)-2-{2-[(2S)-2-amino-5-carbamimidamidop...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180((6S,12S,15S)-1,6-diamino-12-(carboxymethyl)-16-hyd...)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180((6S,12S,15S)-1,6-diamino-12-(carboxymethyl)-16-hyd...)
Affinity DataIC50:  8.20E+4nMAssay Description:Ability of the compound to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180((6S,12S,15S)-1,6-diamino-12-(carboxymethyl)-16-hyd...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50:  1.01E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: >1.65E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: >1.75E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065174((S)-N-((R)-1-Carboxy-3-cyclohexyl-propyl)-3-{2-[et...)
Affinity DataIC50:  1.93E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065166((S)-N-((R)-1-Carbamoyl-2-cyclohexyl-ethyl)-3-{2-[e...)
Affinity DataIC50: >2.35E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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