Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with all data for entry = 50007634
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065797(CHEMBL329488 | Sodium; 8-hydroxy-2-[(E)-2-(3,4,5-t...)
Affinity DataIC50:  260nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065793(8-Hydroxy-2-[(E)-2-(3,4,5-trihydroxy-phenyl)-vinyl...)
Affinity DataIC50:  300nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065793(8-Hydroxy-2-[(E)-2-(3,4,5-trihydroxy-phenyl)-vinyl...)
Affinity DataIC50:  400nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065788((E)-2-(3-carboxy-4-hydroxystyryl)-8-hydroxyquinoli...)
Affinity DataIC50:  600nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065795(CHEMBL100082 | Sodium; 2-[(E)-2-(3,4-dihydroxy-phe...)
Affinity DataIC50:  800nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065796((E)-2-(3,4-dihydroxystyryl)-8-hydroxyquinoline-7-c...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065783(5-(2-{7-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy...)
Affinity DataIC50:  2.20E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065796((E)-2-(3,4-dihydroxystyryl)-8-hydroxyquinoline-7-c...)
Affinity DataIC50:  2.40E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065787(4-(2-(8-hydroxyquinolin-2-yl)vinyl)benzene-1,2-dio...)
Affinity DataIC50:  2.40E+3nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065788((E)-2-(3-carboxy-4-hydroxystyryl)-8-hydroxyquinoli...)
Affinity DataIC50:  2.70E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065790((E)-2-(2,4-dihydroxystyryl)-8-hydroxyquinoline-7-c...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065786(2-[(E)-2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-q...)
Affinity DataIC50:  3.00E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065783(5-(2-{7-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy...)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065790((E)-2-(2,4-dihydroxystyryl)-8-hydroxyquinoline-7-c...)
Affinity DataIC50:  3.70E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065787(4-(2-(8-hydroxyquinolin-2-yl)vinyl)benzene-1,2-dio...)
Affinity DataIC50:  7.40E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065802(Acetic acid 2-acetoxy-5-[(E)-2-(8-acetoxy-quinolin...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065798(Acetic acid 2-((E)-styryl)-quinolin-8-yl ester | A...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065800((E)-3-(3,4-Dihydroxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065784(4-[(E)-2-(8-Nitro-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065784(4-[(E)-2-(8-Nitro-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065799(4-((E)-2-Quinolin-2-yl-vinyl)-benzene-1,2-diol | C...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065791(4-[(E)-2-(8-Amino-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065785(2-Methyl-quinolin-8-ol | CHEMBL316892)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against 3' processing of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065802(Acetic acid 2-acetoxy-5-[(E)-2-(8-acetoxy-quinolin...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065794(8-Hydroxy-2-methyl-quinoline-7-carboxylic acid | 8...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065791(4-[(E)-2-(8-Amino-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065798(Acetic acid 2-((E)-styryl)-quinolin-8-yl ester | A...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065789(2-((E)-Styryl)-quinolin-8-ol | 2-Styryl-quinolin-8...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065800((E)-3-(3,4-Dihydroxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065801(2-[2-(8-hydroxy-2-quinolyl)-(E)-1-ethenyl]-8-quino...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065792((E)-3-(3,4-Dimethoxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065792((E)-3-(3,4-Dimethoxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065789(2-((E)-Styryl)-quinolin-8-ol | 2-Styryl-quinolin-8...)
Affinity DataIC50: >1.00E+5nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065785(2-Methyl-quinolin-8-ol | CHEMBL316892)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50065794(8-Hydroxy-2-methyl-quinoline-7-carboxylic acid | 8...)
Affinity DataIC50:  1.14E+5nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed