Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50007685
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066481((S)-2-Acetylamino-N-[(5S,11R,14S,17R,19aS)-17-cycl...)
Affinity DataIC50:  12nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066483((S)-2-Acetylamino-N-[(5S,12S,15S,18R,20aS)-18-cycl...)
Affinity DataIC50:  90nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066481((S)-2-Acetylamino-N-[(5S,11R,14S,17R,19aS)-17-cycl...)
Affinity DataIC50:  280nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066478((S)-1-[(S)-6-Amino-2-((S)-2-methylamino-3-phenyl-p...)
Affinity DataIC50:  500nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066479((S)-2-[(S)-2-[(R)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  700nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066482((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.80E+3nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066483((S)-2-Acetylamino-N-[(5S,12S,15S,18R,20aS)-18-cycl...)
Affinity DataIC50:  3.20E+3nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066479((S)-2-[(S)-2-[(R)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.10E+4nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066478((S)-1-[(S)-6-Amino-2-((S)-2-methylamino-3-phenyl-p...)
Affinity DataIC50:  1.40E+4nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066482((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.40E+4nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066480((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.44E+5nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066480((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50: >1.00E+6nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50012295(CHEMBL217378 | ISHKDMQLGR | Ile-Ser-His-Lys-Asp-Me...)
Affinity DataIC50: >1.00E+6nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed