Affinity DataIC50: 4.30nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 491nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 3.35E+3nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.76E+3nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 4.11E+3nMAssay Description:relative affinity against dopamine transporter using WIN-35428 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.24E+3nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:relative affinity against serotonin transporter using RTI-55 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:relative affinity against Dopamine receptor D3 in ventral striatum using [3H](+)-7-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+4nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+4nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+4nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:relative affinity against Opioid receptor kappa 1 in insular Ctx using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.72E+4nMAssay Description:relative affinity against Dopamine receptor D2 in striatum using [3H]YM-09151-2 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.45E+4nMAssay Description:Relative affinity against Opioid receptor mu 1 in thalamus using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair