Compile Data Set for Download or QSAR
maximum 50k data
Found 70 Enz. Inhib. hit(s) with all data for entry = 50036679
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068071(CHEMBL2370908 | SRIF)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068063((12S,15R,18S)-9-(4-Amino-butyl)-3-benzyl-15-(4-hyd...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068071(CHEMBL2370908 | SRIF)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068039(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  6nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068043(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068067(1-{3-[(5-Bromo-pyridin-2-yl)-naphthalen-1-ylmethyl...)
Affinity DataKi:  16nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068044(2N-(4-bromobenzyl)-2N-(3-{1-[3-(1H-4-imidazolyl)pr...)
Affinity DataKi:  50nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068066(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  53nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068072(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  70nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068040(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  96nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068056(1-{3-[(4-Bromo-benzyl)-pyridin-2-yl-amino]-propyl}...)
Affinity DataKi:  113nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068055(1-{3-[(4-Bromo-benzyl)-pyridin-2-yl-amino]-propyl}...)
Affinity DataKi:  118nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068045(1-{5-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  132nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068059(1-{2-[(3,4-Dichloro-benzyl)-(5-nitro-pyridin-2-yl)...)
Affinity DataKi:  176nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068058(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  185nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068072(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  310nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068060(4-(1H-Imidazol-4-yl)-piperidine-1-carbothioic acid...)
Affinity DataKi:  413nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068042(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  476nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068064(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  477nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068059(1-{2-[(3,4-Dichloro-benzyl)-(5-nitro-pyridin-2-yl)...)
Affinity DataKi:  500nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068049(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  514nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068047(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  520nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068066(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  565nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068039(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  621nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068045(1-{5-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  777nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068067(1-{3-[(5-Bromo-pyridin-2-yl)-naphthalen-1-ylmethyl...)
Affinity DataKi:  778nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068062(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  803nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068053(1-(4-Amino-butyl)-3-{3-[(5-bromo-pyridin-2-yl)-(3,...)
Affinity DataKi:  830nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068042(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  894nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068060(4-(1H-Imidazol-4-yl)-piperidine-1-carbothioic acid...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068053(1-(4-Amino-butyl)-3-{3-[(5-bromo-pyridin-2-yl)-(3,...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068069(1-(4-Amino-butyl)-3-{3-[(5-bromo-pyridin-2-yl)-nap...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068052(1-(1H-Benzotriazol-5-yl)-3-{2-[(5-bromo-pyridin-2-...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068051(1-(1H-Benzoimidazol-2-ylmethyl)-3-{2-[(5-bromo-pyr...)
Affinity DataKi:  1.20E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068050(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068049(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  1.60E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068047(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068064(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068057(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068061(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  1.90E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068062(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  2.00E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068050(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  2.00E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068040(1-{4-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  2.00E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068069(1-(4-Amino-butyl)-3-{3-[(5-bromo-pyridin-2-yl)-nap...)
Affinity DataKi:  2.00E+3nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068061(1-{3-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)
Affinity DataKi:  2.20E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068065(1-(3-Amino-propyl)-3-{2-[(5-bromo-pyridin-2-yl)-(3...)
Affinity DataKi:  2.30E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068055(1-{3-[(4-Bromo-benzyl)-pyridin-2-yl-amino]-propyl}...)
Affinity DataKi:  2.50E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068052(1-(1H-Benzotriazol-5-yl)-3-{2-[(5-bromo-pyridin-2-...)
Affinity DataKi:  3.00E+3nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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