Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50034984
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.217nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  27nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  30nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50291697((1S,2S,13S)-22-(cyclopropylmethyl)-14-oxa-11,22-di...)
Affinity DataKi:  35nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069179(22-cyclopropylmethyl-16-vinyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  61nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069175(22-cyclopropylmethyl-16-methyl-14-oxa-11,22-diazah...)
Affinity DataKi:  71nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069177(22-cyclopropylmethyl-16-(2-furyl)-14-oxa-11,22-dia...)
Affinity DataKi:  959nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069176(22-cyclopropylmethyl-16-(3-hydroxyphenyl)-14-oxa-1...)
Affinity DataKi:  1.61E+3nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069179(22-cyclopropylmethyl-16-vinyl-14-oxa-11,22-diazahe...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069175(22-cyclopropylmethyl-16-methyl-14-oxa-11,22-diazah...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50291697((1S,2S,13S)-22-(cyclopropylmethyl)-14-oxa-11,22-di...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069181(22-cyclopropylmethyl-16-phenyl-14-oxa-11,22-diazah...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069180(22-cyclopropylmethyl-16-(3-methoxyphenyl)-14-oxa-1...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069176(22-cyclopropylmethyl-16-(3-hydroxyphenyl)-14-oxa-1...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069177(22-cyclopropylmethyl-16-(2-furyl)-14-oxa-11,22-dia...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069180(22-cyclopropylmethyl-16-(3-methoxyphenyl)-14-oxa-1...)
Affinity DataKi: >6.67E+3nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069181(22-cyclopropylmethyl-16-phenyl-14-oxa-11,22-diazah...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069176(22-cyclopropylmethyl-16-(3-hydroxyphenyl)-14-oxa-1...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069180(22-cyclopropylmethyl-16-(3-methoxyphenyl)-14-oxa-1...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069175(22-cyclopropylmethyl-16-methyl-14-oxa-11,22-diazah...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069177(22-cyclopropylmethyl-16-(2-furyl)-14-oxa-11,22-dia...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069181(22-cyclopropylmethyl-16-phenyl-14-oxa-11,22-diazah...)
Affinity DataKi:  1.06E+4nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50291697((1S,2S,13S)-22-(cyclopropylmethyl)-14-oxa-11,22-di...)
Affinity DataKi:  1.09E+4nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069179(22-cyclopropylmethyl-16-vinyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  1.76E+4nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed