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Found 17 Enz. Inhib. hit(s) with all data for entry = 50048431
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50045004(9-fluoro-3-methyl-10-(4-methylpiperazin-1-yl)-7-ox...)
Affinity DataIC50:  4.98E+3nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215357(CHEMBL6353)
Affinity DataIC50:  7.65E+3nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215365(CHEMBL6345)
Affinity DataIC50:  5.32E+4nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215546(CHEMBL268770)
Affinity DataIC50:  1.51E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataIC50:  1.55E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM21691(1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridi...)
Affinity DataIC50:  2.23E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215360(CHEMBL266458)
Affinity DataIC50:  3.07E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215358(CHEMBL204146)
Affinity DataIC50:  3.27E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215366(CHEMBL263076)
Affinity DataIC50:  4.46E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215545(CHEMBL6338)
Affinity DataIC50:  4.99E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215356(CHEMBL6247)
Affinity DataIC50:  5.10E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215364(CHEMBL6335)
Affinity DataIC50:  9.42E+5nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215361(CHEMBL6349)
Affinity DataIC50:  1.50E+6nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215362(CHEMBL6336)
Affinity DataIC50: >1.92E+6nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215363(CHEMBL6365)
Affinity DataIC50: >2.19E+6nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215359(CHEMBL6364)
Affinity DataIC50: >2.19E+6nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50215547(Benzo[C]Chromen-6-One | CHEBI:86511 | CHEMBL6355)
Affinity DataIC50: >2.54E+6nMAssay Description:Inhibition of DNA gyrase supercoiling in Escherichia coli.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed