Affinity DataKi: 1.70nMAssay Description:Compound was evaluated for concentration-dependent and oscillatory increase in [Ca2+], caused by activation of hNK3 receptors in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Bologna
Curated by ChEMBL
University Of Bologna
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Bologna
Curated by ChEMBL
University Of Bologna
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Bologna
Curated by ChEMBL
University Of Bologna
Curated by ChEMBL
Affinity DataKi: 589nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Bologna
Curated by ChEMBL
University Of Bologna
Curated by ChEMBL
Affinity DataKi: 741nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Tested for inhibition of substrate hydrolysis in the presence of porcine kidney esterase at a concentration of 1 uMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University Of Bologna
Curated by ChEMBL
University Of Bologna
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.34E+3nMAssay Description:Compound was evaluated for concentration-dependent and oscillatory increase in [Ca2+], caused by activation of hNK3 receptors in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.32E+3nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair