Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50008217
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071611(6-Azepan-1-ylmethyl-2-(4,4-diphenyl-butyl)-1,2,3,4...)
Affinity DataIC50:  460nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071610(6-Azepan-1-ylmethyl-2-(6,6-diphenyl-hexyl)-1,2,3,4...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071607(6-Azepan-1-ylmethyl-2-[4,4-bis-(4-fluoro-phenyl)-b...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071615(6-Azepan-1-ylmethyl-2-(6,6-diphenyl-hex-5-enyl)-1,...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071612(5-(8-Hydroxy-7-piperidin-1-ylmethyl-isoquinolin-5-...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071616(6-Azepan-1-ylmethyl-2-(5,5-diphenyl-pentyl)-1,2,3,...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071617(6-Azepan-1-ylmethyl-2-[4-(4-fluoro-phenyl)-butyl]-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071614(6-Azepan-1-ylmethyl-2-(3,3-diphenyl-propyl)-1,2,3,...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071608(6-Azepan-1-ylmethyl-2-[4-(4-methoxy-phenyl)-butyl]...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071609(6-Azepan-1-ylmethyl-2-(4-phenyl-butyl)-1,2,3,4-tet...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071618(6-Azepan-1-ylmethyl-isoquinolin-5-ol | CHEMBL78968)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071613(6-Azepan-1-ylmethyl-2-methyl-1,2,3,4-tetrahydro-is...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of N-type calcium channel in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed