Affinity DataKi: 3nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for human Androgen receptor expressed in COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity for human Androgen receptor expressed in COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity towards human glucocorticoid receptor (GR) was determined using [3H]-Dexamethasone as radioligand in SF-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Agonist activity against Human Androgen receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.48E+3nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity against Human Androgen receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.300nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Antagonist activity against Human Androgen receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair