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Found 26 Enz. Inhib. hit(s) with all data for entry = 50008450
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073429(CHEMBL82032 | CHEMBL84575 | N-((S)-1-Carbamimidoyl...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073430(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  41nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073431(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  80nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073429(CHEMBL82032 | CHEMBL84575 | N-((S)-1-Carbamimidoyl...)
Affinity DataIC50:  101nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073426(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  118nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073432(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  135nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073425(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  143nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073428(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  247nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073426(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  333nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073430(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  369nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073431(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  451nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073432(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  627nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50071693(CHEMBL38927 | CVS-1578 | N-((S)-1-Carbamimidoyl-2-...)
Affinity DataIC50:  1.27E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073432(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50:  1.76E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50071693(CHEMBL38927 | CVS-1578 | N-((S)-1-Carbamimidoyl-2-...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073427(CHEMBL331909 | N-((S)-1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073427(CHEMBL331909 | N-((S)-1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073426(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073425(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073430(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073429(CHEMBL82032 | CHEMBL84575 | N-((S)-1-Carbamimidoyl...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073431(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073425(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073428(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073428(2-({(S)-1-[((S)-1-Carbamimidoyl-2-hydroxy-piperidi...)
Affinity DataIC50: >2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against thrombolytic enzyme plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50073427(CHEMBL331909 | N-((S)-1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibitory activity of the compound was evaluated against human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed