Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50008469
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataIC50:  0.0600nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  0.540nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  0.770nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073621(1-(2-Methoxy-phenyl)-4-[3-((S)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50:  1.30nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073614(1-(2-Methoxy-phenyl)-4-[3-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073617(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  2.30nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073620(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  2.40nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073622(2-Dipropylamino-1,2,3,4-tetrahydro-naphthalene-1,8...)
Affinity DataIC50:  2.5nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073610(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  4.30nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073613(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  4.5nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073619(CHEMBL148397 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073615(CHEMBL148234 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033847(CHEMBL108241 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  7.70nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073612(CHEMBL147371 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50052569(CHEMBL107486 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073611(CHEMBL147692 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  34nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073621(1-(2-Methoxy-phenyl)-4-[3-((S)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073616(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((S)-5-m...)
Affinity DataIC50:  89nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073614(1-(2-Methoxy-phenyl)-4-[3-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073618(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((R)-5-m...)
Affinity DataIC50:  320nMAssay Description:In vitro inhibition of [3H]-8-OH-DPAT binding to rat 5-HT 1a receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50033847(CHEMBL108241 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  380nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073617(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073620(1-[3-((S)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073615(CHEMBL148234 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  650nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataIC50:  761nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073618(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((R)-5-m...)
Affinity DataIC50:  870nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073610(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073613(1-[3-((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50052569(CHEMBL107486 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  1.06E+3nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073619(CHEMBL148397 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073611(CHEMBL147692 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073616(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-((S)-5-m...)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50073612(CHEMBL147371 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  3.20E+3nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed