Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 853
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294256(Cis-N-(1-(4-benzyl-3-(methylamino)chroman-6-yl)aze...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294270(US9586945, 21)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294268( trans-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chro...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294267( Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroma...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294266(US9586945, 18b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294265(Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroman...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294264(US9586945, 17b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294263( Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroma...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294262(US9586945, 16b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294261( Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroma...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294260(US9586945, 15b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294259( Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroma...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294256(Cis-N-(1-(4-benzyl-3-(methylamino)chroman-6-yl)aze...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294254(Cis-N-(1-(4-benzyl-3-(methylamino)chroman-6-yl)aze...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294249(Cis-N-(1-(3-(azetidin-1-yl)-4-benzylchroman-6-yl)a...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294244( N-[1-[3-(azetidin-1-yl)-4-benzyl-chroman-6-yl]aze...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294276(Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroman...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294271( Cis-N-(1-(4-benzyl-3-(methylamino)chroman-6-yl)az...)
Affinity DataKi: <10nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294253(Cis-N-(1-(3-(azetidin-1-yl)-4-benzylchroman-6-yl)a...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294258(US9586945, 14b | trans-N-(1-(4-benzyl-7-fluoro-3-(...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294275(Cis-1-(4-benzyl-7-fluoro-6-(3-(5-fluoropyridine-3-...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294255(Cis-N-(1-(-4-benzyl-3-(methylamino)chroman-6-yl)az...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294276(Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroman...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294278(Cis-N-(1-(4-benzyl-3-(propylamino)chroman-6-yl)aze...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294279(Cis-N-(1-(4-benzyl-3-(diethylamino)chroman-6-yl)az...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294250(Cis-N-(1-(3-(azetidin-1-yl)-4-benzyl-7-fluorochrom...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294257(Cis-N-(1-(4-benzyl-7-fluoro-3-(methylamino)chroman...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294248(Cis-N-(1-(3-(azetidin-1-yl)-4-benzylchroman-6-yl)a...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294247(Cis-N-(1-(3-(azetidin-1-yl)-4-benzylchroman-6-yl)a...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294246(Cis-N-(1-(3-(azetidin-1-yl)-4-benzylchroman-6-yl)a...)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294269(US9586945, 20)
Affinity DataKi: <100nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294281( Cis-N-(1-(4-benzyl-3-(cyclobutylamino)chroman-6-y...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294274(Cis-N-(1-(4-benzyl-3-(methylamino)chroman-6-yl)aze...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294245(Cis-N-(1-(3-(azetidin-1-yl)-4-benzylchroman-6-yl)a...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294280(Cis-N-(1-(4-benzyl-3-((cyclopropylmethyl)amino)chr...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294251(Cis-N-(1-(3-(azetidin-1-yl)-4-benzyl-7-fluorochrom...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294271( Cis-N-(1-(4-benzyl-3-(methylamino)chroman-6-yl)az...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Abbvie Deutschland

US Patent
LigandPNGBDBM294252(Cis-N-(1-(3-(azetidin-1-yl)-4-benzyl-7-fluorochrom...)
Affinity DataKi: <1.00E+3nMAssay Description:1. [3H]-Glycine uptake into recombinant CHO cells expressing human GlyT1: Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent