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Found 232 Enz. Inhib. hit(s) with all data for entry = 5786
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)
Affinity DataIC50: >205nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93514((3Z,5Z)-3,5-bis(3,4-dichlorobenzylidene)-1-(3-morp...)
Affinity DataIC50: >614nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM67266(4-chloranyl-1-ethyl-3-nitro-quinolin-2-one | 4-chl...)
Affinity DataIC50:  622nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM80083(3'-ketospiro[1,3-dithiole-2,7'-dithiolo[4,3-b]thio...)
Affinity DataIC50:  727nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM88687(4-(keto-methyl-oxido-sulfuraniumyl)-3-nitro-benzoi...)
Affinity DataIC50:  800nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM58440(2-[[5-(2-ethyl-5-methyl-3-pyrazolyl)-4-methyl-1,2,...)
Affinity DataIC50:  802nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM41585((E)-4,4-dimethyl-1-(3-nitrophenyl)-2-(1,2,4-triazo...)
Affinity DataIC50:  852nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM68076(4,5-bis(chloranyl)-2-[6-(2-methylphenoxy)pyrimidin...)
Affinity DataIC50:  882nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM41609((4,5-dichloro-6-oxopyridazin-1-yl)methyl 4-methylb...)
Affinity DataIC50:  889nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM54804(2-[1-[(Z)-1-(4-bromobenzoyl)-2-(2-furyl)vinyl]-2-p...)
Affinity DataIC50:  895nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM46457((Z)-4,4-Dimethyl-1-(3-nitro-phenyl)-2-[1,2,4]triaz...)
Affinity DataIC50:  897nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93528((1S,4R,6S,6aR,9R,11bS)-methyl 1-acetoxy-6-hydroxy-...)
Affinity DataIC50:  917nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81246((3E,5E)-1,1-diketo-3,5-bis(4-nitrobenzylidene)thia...)
Affinity DataIC50:  930nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM60237(2-[1-[(Z)-1-(2-furanyl)-3-oxo-3-(4-phenylphenyl)pr...)
Affinity DataIC50:  945nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM34180(3-(3,4-dimethoxyphenyl)-1-[(pentafluorophenyl)sulf...)
Affinity DataIC50:  951nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM59054(4-[(7-chloranyl-4-nitro-1,3-dihydro-2,1,3-benzoxad...)
Affinity DataIC50:  969nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM53797(2-[1-[(Z)-1-(2-furanyl)-3-oxo-3-phenylprop-1-en-2-...)
Affinity DataIC50:  1.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM61664(1-anilino-3-(4-chlorophenyl)-1H-pyrrole-2,5-dione ...)
Affinity DataIC50:  1.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93512(4-keto-1,3-diphenyl-6-(2-pyrrolidinoethylthio)-2-t...)
Affinity DataIC50:  1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM71504(1-(5-chlorobenzofurazan-4-yl)sulfonylisonipecotic ...)
Affinity DataIC50:  1.12E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM42532(2-[1-[(Z)-1-(4-chlorobenzoyl)-2-(2-furyl)vinyl]-2-...)
Affinity DataIC50:  1.13E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM71379(3,4-bis(chloranyl)-6-phenyl-pyran-2-one | 3,4-dich...)
Affinity DataIC50:  1.15E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM68080(4,5-bis(bromanyl)-2-(4,6-dimethoxypyrimidin-2-yl)p...)
Affinity DataIC50:  1.18E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM83275(MLS002701540 | SMR001565141 | cid_457901)
Affinity DataIC50:  1.19E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM80085(10-(diiodomethylene)phenanthren-9-one | 10-(diiodo...)
Affinity DataIC50:  1.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM80701(2-(1,4-diketo-2-naphthyl)-2-methyl-propionaldehyde...)
Affinity DataIC50:  1.23E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM77570(3-[(5-nitro-1,3-thiazol-2-yl)sulfanyl]-4-prop-2-en...)
Affinity DataIC50:  1.32E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93522(2-[4-morpholinyl(phenyl)methylidene]-3H-inden-1-on...)
Affinity DataIC50:  1.35E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM67158(9-(2,4-dihydroxyphenyl)-3,3,6,6-tetramethyl-4,5,7,...)
Affinity DataIC50:  1.36E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93505(MLS002701772 | SMR001565366 | cid_3795051)
Affinity DataIC50:  1.36E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM60990(MLS001336050 | SMR000875330 | Thime-rosal | Thimer...)
Affinity DataIC50:  1.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93533((6aR,11aS)-9-chloro-6-cyclohexyl-5-keto-6a,11-dihy...)
Affinity DataIC50:  1.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM72932((5Z)-5-(4-chloro-3-nitro-benzylidene)-3-[2-(dimeth...)
Affinity DataIC50:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93466(1-(4-fluoranyl-3-nitro-phenyl)sulfonylazepane | 1-...)
Affinity DataIC50:  1.53E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM33080(2-[[7-(1,3-benzothiazol-2-ylsulfanyl)-4-nitro-2,1,...)
Affinity DataIC50:  1.54E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM65997((4Z)-3-methyl-4-[(1-phenyl-3-thiophen-2-yl-4-pyraz...)
Affinity DataIC50:  1.55E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93478((3Z)-3-[(3Z)-2-keto-3-(2-ketoindolin-3-ylidene)pro...)
Affinity DataIC50:  1.55E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93542((6aR,11aS)-6-cyclohexyl-3-methoxy-9-methyl-5-oxo-6...)
Affinity DataIC50:  1.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93493(MLS001099311 | N-[2-[(5Z)-5-(4-chloro-3-nitro-benz...)
Affinity DataIC50:  1.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93507(MLS002701874 | SMR001565464 | cid_341502)
Affinity DataIC50:  1.63E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM79544(1-[1-(4-methoxyphenyl)-2-nitro-ethyl]-3,5-dimethyl...)
Affinity DataIC50:  1.63E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM54724(1-anilino-3-phenyl-1H-pyrrole-2,5-dione | 1-anilin...)
Affinity DataIC50:  1.68E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM72561(1-(4-methylanilino)-3-phenylpyrrole-2,5-dione | 1-...)
Affinity DataIC50:  1.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM48011(1-benzyl-5-[(E)-2-nitroethenyl]indole | 1-benzyl-5...)
Affinity DataIC50:  1.74E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50164(1-ethoxy-4-(2-nitrovinyl)naphthalene | 1-ethoxy-4-...)
Affinity DataIC50:  1.76E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM65213(4-[[2-(4,5-dichloro-6-keto-pyridazin-1-yl)acetyl]a...)
Affinity DataIC50:  1.77E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM42060(4,5-bis(chloranyl)-2-[2-(4-naphthalen-2-ylsulfonyl...)
Affinity DataIC50:  1.77E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM61011((3'S,4'R)-1'-(4-chlorophenyl)-2'-cyano-spiro[fluor...)
Affinity DataIC50:  1.78E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM66727(3-pyridinecarboxylic acid [2-methoxy-4-[(E)-2-nitr...)
Affinity DataIC50:  1.82E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM93467(2-(4-brosylpiperazino)-N-[(E)-(4-chloro-3-nitro-be...)
Affinity DataIC50:  1.83E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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