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Target
fMet-Leu-Phe receptor
Ligand
BDBM37772
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki
5500±n/a nM
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
fMet-Leu-Phe receptor
Synonyms:
FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38456.14
Organism:
Homo sapiens (Human)
Description:
gi_4503779
Residue:
350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVTTISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIALDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNFSPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPLRVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPMLYVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
  
Inhibitor
Name:
BDBM37772
Synonyms:
2-(benzylsulfonyl)-N,N-diisobutylacetamide | 2-benzylsulfonyl-N,N-bis(2-methylpropyl)acetamide | 2-benzylsulfonyl-N,N-diisobutyl-acetamide | MLS000050849 | N,N-bis(2-methylpropyl)-2-(phenylmethyl)sulfonyl-ethanamide | N,N-bis(2-methylpropyl)-2-(phenylmethyl)sulfonylacetamide | SMR000078536 | cid_2218678
Type:
Small organic molecule
Emp. Form.:
C17H27NO3S
Mol. Mass.:
325.466
SMILES:
CC(C)CN(CC(C)C)C(=O)CS(=O)(=O)Cc1ccccc1
Structure:
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