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Target
Zinc finger protein mex-5
Ligand
BDBM52464
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52464
Synonyms:
(3Z)-3-(2-keto-4-methyl-pentylidene)-6-methyl-4H-1,4-benzoxazin-2-one | (3Z)-6-methyl-3-(4-methyl-2-oxidanylidene-pentylidene)-4H-1,4-benzoxazin-2-one | (3Z)-6-methyl-3-(4-methyl-2-oxopentylidene)-4H-1,4-benzoxazin-2-one | 6-Methyl-3-[4-methyl-2-oxo-pent-(E)-ylidene]-3,4-dihydro-benzo[1,4]oxazin-2-one | MLS000588162 | SMR000220136 | cid_6888034
Type:
Small organic molecule
Emp. Form.:
C15H17NO3
Mol. Mass.:
259.3004
SMILES:
CC(C)CC(=O)Cc1nc2cc(C)ccc2oc1=O
Structure:
Search PDB for entries with ligand similarity: