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Target
Zinc finger protein mex-5
Ligand
BDBM52471
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52471
Synonyms:
2-(1-adamantyl)-N-(1-iminoisoindolin-2-yl)acetamide | 2-(1-adamantyl)-N-(3-azanylidene-1H-isoindol-2-yl)ethanamide | 2-(1-adamantyl)-N-(3-imino-1H-isoindol-2-yl)acetamide | MLS000402247 | SMR000263874 | cid_4308688
Type:
Small organic molecule
Emp. Form.:
C20H25N3O
Mol. Mass.:
323.432
SMILES:
[H]C12CC3([H])CC([H])(C1)CC(CC(=O)NN1Cc4ccccc4C1=N)(C2)C3 |TLB:8:6:26:1.25.2,8:1:26:6.9.5,THB:2:1:9:3.26.5|
Structure:
Search PDB for entries with ligand similarity: