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Target
Bcl-2-like protein 11
Ligand
BDBM67038
Substrate
n/a
Meas. Tech.
Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis
EC50
>350000±n/a nM
Citation
 PubChem, PC Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis PubChem Bioassay (2010)[AID] 
Target
Name:
Bcl-2-like protein 11
Synonyms:
B2L11_HUMAN | BCL2-like 11 isoform 1 | BCL2L11 | BIM
Type:
PROTEIN
Mol. Mass.:
22175.26
Organism:
Homo sapiens (Human)
Description:
EBI_101325
Residue:
198
Sequence:
MAKQPSDVSSECDREGRQLQPAERPPQLRPGAPTSLQTEPQGNPEGNHGGEGDSCPHGSPQGPLAPPASPGPFATRSPLFIFMRRSSLLSRSSSGYFSFDTDRSPAPMSCDKSTQTPSPPCQAFNHYLSAMASMRQAEPADMRPEIWIAQELRRIGDEFNAYYARRVFLNNYQAAEDHPRMVILRLLRYIVRLVWRMH
  
Inhibitor
Name:
BDBM67038
Synonyms:
MLS002302624 | N-cyclopentyl-9,10,10-triketo-6-m-cumenyl-thioxanthene-1-carboxamide | N-cyclopentyl-9,10,10-trioxo-6-(3-propan-2-ylphenyl)-1-thioxanthenecarboxamide | N-cyclopentyl-9,10,10-trioxo-6-(3-propan-2-ylphenyl)thioxanthene-1-carboxamide | N-cyclopentyl-9,10,10-tris(oxidanylidene)-6-(3-propan-2-ylphenyl)thioxanthene-1-carboxamide | SMR001318652 | cid_44143835
Type:
Small organic molecule
Emp. Form.:
C28H27NO4S
Mol. Mass.:
473.583
SMILES:
CC(C)c1cccc(c1)-c1ccc2C(=O)c3c(cccc3S(=O)(=O)c2c1)C(=O)NC1CCCC1
Structure:
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