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Reaction Details
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TargetCannabinoid receptor 2
LigandBDBM68301
Substrate/Competitorn/a
Meas. Tech.SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2
IC50>32000±n/a nM
Citation PubChem, PC SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:39690.94
Organism:Homo sapiens (Human)
Description:P34972
Residue:360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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  Blast E-value cutoff:
BDBM68301
NameBDBM68301
Synonyms:4-(difluoromethoxy)-N-(2-methoxy-5-morpholin-4-ylsulfonylphenyl)benzamide | 4-(difluoromethoxy)-N-(2-methoxy-5-morpholinosulfonyl-phenyl)benzamide | 4-(difluoromethoxy)-N-[2-methoxy-5-(4-morpholinylsulfonyl)phenyl]benzamide | 4-[bis(fluoranyl)methoxy]-N-(2-methoxy-5-morpholin-4-ylsulfonyl-phenyl)benzamide | MLS-0405205.0001 | cid_4676506
TypeSmall organic molecule
Emp. Form.C19H20F2N2O6S
Mol. Mass.442.434
SMILESCOc1ccc(cc1NC(=O)c1ccc(OC(F)F)cc1)S(=O)(=O)N1CCOCC1
Structure
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n/a