Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetADRA2C
LigandBDBM81815
Substrate/Competitorn/a
Ki 0.14±n/a nM
CommentsPDSP_1049
Citation Blaxall, HSMurphy, TJBaker, JCRay, CBylund, DB Characterization of the alpha-2C adrenergic receptor subtype in the opossum kidney and in the OK cell line. J Pharmacol Exp Ther259:323-9 (1991) [PubMed]
More Info.:Get all data from this article
 
ADRA2C
Name:ADRA2C
Synonyms:adrenergic Alpha2C
Type:Enzyme Catalytic Domain
Mol. Mass.:27257.01
Organism:OK
Description:adrenergic Alpha2C ADRA2C OK::G3GWB4
Residue:230
Sequence:
MAYWYFGQVWCGVYLALDVLFCTSSIVHLCAISLDRYWSVTQAVEYNLKRTPRRVKATIV
AVWLISAVISFPPLVSFYRRSDGAAYPQCGLNDETWYILSSCIGSFFAPCLIMGLVYARI
YRFFLSRRRRARSSVCRRKVAQAREKRFTFVLAVVMGVFVLCWFPFFFSYSLYGICREAC
QLPEPLFKFFFWIGYCKSSLNPVIYTVFNQDFRRSFKHILFRRRRRGFRQ
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM81815
NameBDBM81815
Synonyms:CAS_196343 | L-654,284 | NSC_196343
TypeSmall organic molecule
Emp. Form.C46H67N9O9S2
Mol. Mass.954.209
SMILESCCOc1ccc(CC(NC(=O)CC2(S)CCCCC2)C(=O)NC(Cc2ccccc2)C(=O)NC(C(C)C)C(=O)NC(CC(N)=O)C(=O)NC(C=S)C(=O)NC(CCCCN)C(N)=O)cc1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a