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Target
Voltage-dependent calcium channel gamma-1 subunit
Ligand
BDBM81818
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_2651
Citation
 Garritsen, A; Ijzerman, AP; Tulp, MT; Cragoe, EJ; Soudijn, W Receptor binding profiles of amiloride analogues provide no evidence for a link between receptors and the Na+/H+ exchanger, but indicate a common structure on receptor proteins. J Recept Res 11:891-907 (1991) [PubMed]  Article 
Target
Name:
Voltage-dependent calcium channel gamma-1 subunit
Synonyms:
CACNG1 | CACNLG | CCG1_HUMAN | Calcium channel (DHP) | Voltage-dependent calcium channel gamma-1 subunit
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25030.69
Organism:
Homo sapiens (Human)
Description:
Calcium channel (DHP) 0 0::Q06432
Residue:
222
Sequence:
MSQTKMLKVRVTLFCILAGIVLAMTAVVTDHWAVLSPHMEHHNTTCEAAHFGLWRICTKRIPMDDSKTCGPITLPGEKNCSYFRHFNPGESSEIFEFTTQKEYSISAAAIAIFSLGFIILGSLCVLLSLGKKRDYLLRPASMFYAFAGLCILVSVEVMRQSVKRMIDSEDTVWIEYYYSWSFACACAAFILLFLGGLALLLFSLPRMPRNPWESCMDAEPEH
  
Inhibitor
Name:
BDBM81818
Synonyms:
CAS_1794 | CHEMBL1909810 | HMA | NSC_1794
Type:
Small organic molecule
Emp. Form.:
C12H18ClN7O
Mol. Mass.:
311.771
SMILES:
NC(=N)NC(=O)c1nc(Cl)c(nc1N)N1CCCCCC1
Structure:
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