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TargetCCKBR
LigandBDBM81869
Substrate/Competitorn/a
Ki 510±n/a nM
CommentsPDSP_2194
Citation Lin, CWShiosaki, KMiller, TRWitte, DGBianchi, BRWolfram, CAKopecka, HCraig, RWagenaar, FNadzan, AM Characterization of two novel cholecystokinin tetrapeptide (30-33) analogues, A-71623 and A-70874, that exhibit high potency and selectivity for cholecystokinin-A receptors. Mol Pharmacol39:346-51 (1991) [PubMed]
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CCKBR
Name:CCKBR
Synonyms:Cholecystokinin A
Type:Enzyme Catalytic Domain
Mol. Mass.:48683.10
Organism:GUINEA PIG
Description:Cholecystokinin A CCKBR GUINEA PIG::H0VZC5
Residue:450
Sequence:
MELLKLNRSLQGPGPGPGAPLCRPAGPLLNSSGAGNVSCETPRIRGAGTRVKSMAILFNV
TSLLSCWNKYRIIKVLGLSRRLRTVTKAFLLSLAVSDLLLAVACMPFTLLPNLMGTFIFG
TVICKAVSYLMGVSVSVSTLSLVAIALERYSAICRPLQARVWQTRSHAARVILATWLLSG
LLMVPYPVYTAVQPVGPRVLQCVHRWPNARVRQTWSVLLLLLLFFVPGVVMAVAYGLISR
ELYLGLRFDGDADSESQSRVRGPGGLSGSAPGPAHQNGRCRPESGLSGEDSDGCYVQLPR
SRPALELSALAASTPAPGPGPRPTQAKLLAKKRVVRMLLVIVVLFFLCWLPVYSANTWRA
FDGPGAHRALSGAPISFIHLLSYASACVNPLVYCFMHRRFRQACLDTCARCCPRPPRARP
RPLPEEDPPTPSIASLSRLSYTTISTLGPG
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BDBM81869
NameBDBM81869
Synonyms:A-57282
Typen/a
Emp. Form.C43H53N7O10
Mol. Mass.827.9218
SMILESCC(C)(C)OC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)N(C(=O)C(N)Cc1ccccc1)C(=O)C(CC(O)=O)NC(=O)C(N)CCCCNC(=O)OCc1ccccc1
Structure
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