Reaction Details Report a problem with these data
Target
Cholecystokinin
Ligand
BDBM50005459
Substrate
n/a
Ki
22±n/a nM
Comments
PDSP_2217
Citation
 Lotti, VJ; Chang, RS A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260. Eur J Pharmacol 162:273-80 (1989) [PubMed]  Article 
Target
Name:
Cholecystokinin
Synonyms:
CCK | CCKN_PIG | Cholecystokinin B
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12528.64
Organism:
GUINEA PIG
Description:
Cholecystokinin B 0 GUINEA PIG::P01356
Residue:
114
Sequence:
MNGGLCLCVLMAVLAAGTLAQPVPPADSAVPGAQEEEAHRRQLRAVQKVDGESRAHLGALLARYIQQARKAPSGRVSMIKNLQSLDPSHRISDRDYMGWMDFGRRSAEEYEYTS
  
Inhibitor
Name:
BDBM50005459
Synonyms:
4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-butyric acid | CHEMBL9485 | CR 1409
Type:
Small organic molecule
Emp. Form.:
C22H32Cl2N2O4
Mol. Mass.:
459.406
SMILES:
CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Structure:
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