Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM81989
Substrate
n/a
Ki
6.6±n/a nM
Comments
PDSP_3143
Citation
 Shank, RP; Vaught, JL; Pelley, KA; Setler, PE; McComsey, DF; Maryanoff, BE McN-5652: a highly potent inhibitor of serotonin uptake. J Pharmacol Exp Ther 247:1032-8 (1988) [PubMed] 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM81989
Synonyms:
CAS_68717 | Clovoxamine | NSC_68717
Type:
Small organic molecule
Emp. Form.:
C14H21ClN2O2
Mol. Mass.:
284.782
SMILES:
COCCCCC(=NOCCN)c1ccc(Cl)cc1 |w:7.7|
Structure:
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