Target
Cholecystokinin
Ligand
BDBM81963
Substrate
n/a
Ki
3.3±n/a nM
Comments
PDSP_2672
Citation
 Van Dijk, ARichards, JGTrzeciak, AGillessen, DMöhler, H Cholecystokinin receptors: biochemical demonstration and autoradiographical localization in rat brain and pancreas using [3H] cholecystokinin8 as radioligand. J Neurosci 4:1021-33 (1984) [PubMed] 
Target
Name:
Cholecystokinin
Synonyms:
CCKN_RAT | Cck
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12844.29
Organism:
RAT
Description:
Cholecystokinin 0 RAT::P01355
Residue:
115
Sequence:
MKCGVCLCVVMAVLAAGALAQPVVPVEAVDPMEQRAEEAPRRQLRAVLRPDSEPRARLGALLARYIQQVRKAPSGRMSVLKNLQGLDPSHRISDRDYMGWMDFGRRSAEDYEYPS
  
Inhibitor
Name:
BDBM81963
Synonyms:
CAS_9011-97-6 | CCK | CCK33 | CHOLECYSTOKININ
Type:
Small organic molecule
Emp. Form.:
C166H261N51O52S4
Mol. Mass.:
3931.419
SMILES:
n/a
Structure:
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