Reaction Details Report a problem with these data
Target
Cholecystokinin
Ligand
BDBM81330
Substrate
n/a
Ki
0.35±n/a nM
Comments
PDSP_2615
Citation
 Van Dijk, A; Richards, JG; Trzeciak, A; Gillessen, D; Möhler, H Cholecystokinin receptors: biochemical demonstration and autoradiographical localization in rat brain and pancreas using [3H] cholecystokinin8 as radioligand. J Neurosci 4:1021-33 (1984) [PubMed] 
Target
Name:
Cholecystokinin
Synonyms:
CCKN_RAT | Cck
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12844.29
Organism:
RAT
Description:
Cholecystokinin 0 RAT::P01355
Residue:
115
Sequence:
MKCGVCLCVVMAVLAAGALAQPVVPVEAVDPMEQRAEEAPRRQLRAVLRPDSEPRARLGALLARYIQQVRKAPSGRMSVLKNLQGLDPSHRISDRDYMGWMDFGRRSAEDYEYPS
  
Inhibitor
Name:
BDBM81330
Synonyms:
+ 1 mM GTP | GTP
Type:
Small organic molecule
Emp. Form.:
C10H13N5O14P3
Mol. Mass.:
520.1583
SMILES:
Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H](COP([O-])(=O)OP([O-])(=O)OP(O)([O-])=O)C(O)C1O |r|
Structure:
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