Reaction Details
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Report a problem with these dataTarget
Somatostatin receptor type 4
Ligand
BDBM82257
Substrate
n/a
Ki
1.2±n/a nM
Comments
PDSP_3339
Citation
Rossowski, WJ; Gu, ZF; Akarca, US; Jensen, RT; Coy, DH Characterization of somatostatin receptor subtypes controlling rat gastric acid and pancreatic amylase release. Peptides 15:1421-4 (1994) [PubMed] Article More Info.:
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SSR4_RAT | Somatostatin receptor | Somatostatin receptor type 4 | Sstr4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42096.84
Organism:
RAT
Description:
SOMATOSTATIN SST4 SSTR4 RAT::P30937
Residue:
384
Sequence:
MNTPATLPLGGEDTTWTPGINASWAPDEEEDAVRSDGTGTAGMVTIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASAAALRHWPFGAVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAVFADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGPGCICPPLPCQQEPMQAEPACKRVPFTKTTTF
Inhibitor
Name:
BDBM82257
Synonyms:
D-Phe-Phe-Tyr-D-Trp-Lys-Val-Phe-Thr-NH2 | DC-25-12
Type:
n/a
Emp. Form.:
C61H75N11O10
Mol. Mass.:
1122.3159
SMILES:
CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)C(N)c1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O
Structure:
