Reaction Details
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Report a problem with these dataTarget
Somatostatin receptor type 5
Ligand
BDBM82256
Substrate
n/a
Ki
158±n/a nM
Comments
PDSP_3341
Citation
Rossowski, WJ; Gu, ZF; Akarca, US; Jensen, RT; Coy, DH Characterization of somatostatin receptor subtypes controlling rat gastric acid and pancreatic amylase release. Peptides 15:1421-4 (1994) [PubMed] Article More Info.:
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SSR5_RAT | Somatostatin receptor | Somatostatin receptor type 5 | Sstr5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39986.50
Organism:
RAT
Description:
SOMATOSTATIN SST5 SSTR5 RAT::P30938
Residue:
363
Sequence:
MEPLSLASTPSWNASAASSGNHNWSLVGSASPMGARAVLVPVLYLLVCTVGLSGNTLVIYVVLRHAKMKTVTNVYILNLAVADVLFMLGLPFLATQNAVVSYWPFGSFLCRLVMTLDGINQFTSIFCLMVMSVDRYLAVVHPLRSARWRRPRVAKMASAAVWVFSLLMSLPLLVFADVQEGWGTCNLSWPEPVGLWGAAFITYTSVLGFFGPLLVICLCYLLIVVKVKAAGMRVGSSRRRRSEPKVTRMVVVVVLVFVGCWLPFFIVNIVNLAFTLPEEPTSAGLYFFVVVLSYANSCANPLLYGFLSDNFRQSFRKVLCLRRGYGMEDADAIEPRPDKSGRPQATLPTRSCEANGLMQTSRI
Inhibitor
Name:
BDBM82256
Synonyms:
BIM 23056 | CAS_150155-61-6 | D-Phe-Phe-Tyr-D-Trp-Lys-Val-Phe-D-Nal-NH2 | DC-25-20
Type:
Small organic molecule
Emp. Form.:
C71H81N11O9
Mol. Mass.:
1232.4711
SMILES:
CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](N)Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](Cc1ccc2ccccc2c1)C(N)=O |r|
Structure:
