Target
Neuropeptide Y receptor type 1
Ligand
BDBM82299
Substrate
n/a
Ki
0.14±n/a nM
Comments
PDSP_1558
Citation
 Gerald, CAdham, NKao, HTOlsen, MALaz, TMSchechter, LEBard, JAVaysse, PJHartig, PRBranchek, TA The 5-HT4 receptor: molecular cloning and pharmacological characterization of two splice variants. EMBO J 14:2806-15 (1995) [PubMed] 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44399.07
Organism:
Homo sapiens (Human)
Description:
NPY-Y1 NPY1R HUMAN::P25929
Residue:
384
Sequence:
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMTDEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKINNNDDNEKI
  
Inhibitor
Name:
BDBM82299
Synonyms:
PYY Pro34, Human
Type:
Small organic molecule
Emp. Form.:
C194H293N53O57
Mol. Mass.:
4279.7231
SMILES:
n/a
Structure:
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