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Target
Somatostatin receptor type 2
Ligand
BDBM82457
Substrate
n/a
Ki
83.17±n/a nM
Comments
PDSP_1032
Citation
 Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol 350:441-53 (1994) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 2
Synonyms:
SOMATOSTATIN SST2 | SSR2_MOUSE | Smstr2 | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sst2 | Sstr2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41234.26
Organism:
MOUSE
Description:
SOMATOSTATIN SST2 SSTR2 MOUSE::P30875
Residue:
369
Sequence:
MEMSSEQLNGSQVWVSSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCGNTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMTVDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWCVSLLVILPIMIYAGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGIRVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVILTYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTEDGERSDSKQDKSRLNETTETQRTLLNGDLQTSI
  
Inhibitor
Name:
BDBM82457
Synonyms:
(1R,4S,7S,10R,13S,16R)-4-[(R)-1-Hydroxyethyl]-7-(4-aminobutyl)-10-(1H-indole-3-ylmethyl)-13-benzyl-28,29-dithia-2,5,8,11,14,17,25-heptaazabicyclo[14.10.4]triacontane-3,6,9,12,15,18,26-heptone | L-362,823
Type:
Small organic molecule
Emp. Form.:
C43H59N9O8S2
Mol. Mass.:
894.114
SMILES:
C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H]2CSSC[C@H](NC1=O)C(=O)NCCCCCCC(=O)N2
Structure:
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