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Target
5-hydroxytryptamine receptor 1B
Ligand
BDBM81499
Substrate
n/a
Ki
2.51±n/a nM
Comments
PDSP_596
Citation
 Boess, FG; Martin, IL Molecular biology of 5-HT receptors. Neuropharmacology 33:275-317 (1994) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 1B
Synonyms:
5-HT1B | 5-hydroxytryptamine receptor 1B (5HT1B) | 5HT1B_MOUSE | 5ht1b | Htr1b
Type:
Enzyme
Mol. Mass.:
43090.29
Organism:
Mus musculus (Mouse)
Description:
P28334
Residue:
386
Sequence:
MEEQGIQCAPPPPAASQTGVPLTNLSHNCSADGYIYQDSIALPWKVLLVALLALITLATTLSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPISTMYTVTGRWTLGQVVCDFWLSSDITCCTASIMHLCVIALDRYWAITDAVEYSAKRTPKRAAIMIVLVWVFSISISLPPFFWRQAKAEEEMLDCFVNTDHVLYTVYSTVGAFYLPTLLLIALYGRIYVEARSRILKQTPNKTGKRLTRAQLITDSPGSTSSVTSINSRAPDVPSESGSPVYVNQVKVRVSDALLEKKKLMAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHMAIFDFFNWLGYLNSLINPIIYTMSNEDFKQAFHKLIRFKCAG
  
Inhibitor
Name:
BDBM81499
Synonyms:
CAS_155346 | CYANOPINDOLOL | CYANOPINDOLOL(+/-) | NSC_155346
Type:
Small organic molecule
Emp. Form.:
C16H21N3O2
Mol. Mass.:
287.3568
SMILES:
CC(C)(C)NCC(O)COc1cccc2[nH]c(cc12)C#N
Structure:
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