Reaction Details Report a problem with these data
Target
Somatostatin receptor type 4
Ligand
BDBM84641
Substrate
n/a
Ki
50±n/a nM
Comments
PDSP_1946
Citation
 Raynor, K; O'Carroll, AM; Kong, H; Yasuda, K; Mahan, LC; Bell, GI; Reisine, T Characterization of cloned somatostatin receptors SSTR4 and SSTR5. Mol Pharmacol 44:385-92 (1993) [PubMed] 
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SSR4_RAT | Somatostatin receptor | Somatostatin receptor type 4 | Sstr4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42096.84
Organism:
RAT
Description:
SOMATOSTATIN SST4 SSTR4 RAT::P30937
Residue:
384
Sequence:
MNTPATLPLGGEDTTWTPGINASWAPDEEEDAVRSDGTGTAGMVTIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASAAALRHWPFGAVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAVFADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGPGCICPPLPCQQEPMQAEPACKRVPFTKTTTF
  
Inhibitor
Name:
BDBM84641
Synonyms:
SA V | c[Aoc-Phe-D-Trp-Lys-Thr(Bzl)]
Type:
Small organic molecule
Emp. Form.:
C46H62N8O6
Mol. Mass.:
823.0345
SMILES:
CC(OCc1ccccc1)C1NC(=O)C(CCCCCCCCN)NC(=O)C(Cc2ccccc2)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(CCCN)NC1=O
Structure:
Search PDB for entries with ligand similarity: