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Target
Cholecystokinin receptor type A
Ligand
BDBM50005470
Substrate
n/a
Meas. Tech.
ChEBML_47649
Ki
450±n/a nM
Citation
 van der Bent, A; Blommaert, AG; Melman, CT; IJzerman, AP; van Wijngaarden, I; Soudijn, W Hybrid cholecystokinin-A antagonists based on molecular modeling of lorglumide and L-364,718. J Med Chem 35:1042-9 (1992) [PubMed]  Article 
Target
Name:
Cholecystokinin receptor type A
Synonyms:
CCKAR_RAT | Cckar | Cholecystokinin peripheral | Cholecystokinin receptor | Cholecystokinin receptor type A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49676.37
Organism:
RAT
Description:
Cholecystokinin central 0 RAT::P30551
Residue:
444
Sequence:
MSHSPARQHLVESSRMDVVDSLLMNGSNITPPCELGLENETLFCLDQPQPSKEWQSALQILLYSIIFLLSVLGNTLVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPNLLKDFIFGSAVCKTTTYFMGTSVSVSTFNLVAISLERYGAICRPLQSRVWQTKSHALKVIAATWCLSFTIMTPYPIYSNLVPFTKNNNQTANMCRFLLPSDAMQQSWQTFLLLILFLLPGIVMVVAYGLISLELYQGIKFDASQKKSAKEKKPSTGSSTRYEDSDGCYLQKSRPPRKLELQQLSSGSGGSRLNRIRSSSSAANLIAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAEKHLSGTPISFILLLSYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGPPGVRGEVGEEEDGRTIRALLSRYSYSHMSTSAPPP
  
Inhibitor
Name:
BDBM50005470
Synonyms:
CHEMBL8949 | Naphthalene-2-carboxylic acid (3,3-diphenyl-allyl)-amide
Type:
Small organic molecule
Emp. Form.:
C26H21NO
Mol. Mass.:
363.451
SMILES:
O=[#6](-[#7]-[#6]\[#6]=[#6](/c1ccccc1)-c1ccccc1)-c1ccc2ccccc2c1
Structure:
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